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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference | 
|---|---|---|---|---|---|---|---|---|
| Nav1.7 in Human [GtoPdb: 584] [UniProtKB: Q15858] | ||||||||
| GtoPdb | - | - | 5.15 | pIC50 | 7100 | nM | IC50 | Biochem Biophys Res Commun (2024) 721: 150126 [PMID:38776832] | 
| Nav1.8 in Human [GtoPdb: 585] [UniProtKB: Q9Y5Y9] | ||||||||
| GtoPdb | - | - | 4.94 | pIC50 | 11400 | nM | IC50 | Biochem Biophys Res Commun (2024) 721: 150126 [PMID:38776832] | 
| Nav1.9 in Human [GtoPdb: 586] [UniProtKB: Q9UI33] | ||||||||
| GtoPdb | - | - | 5.17 | pIC50 | 6700 | nM | IC50 | Biochem Biophys Res Commun (2024) 721: 150126 [PMID:38776832] | 
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.