RJG-2051 [Ligand Id: 13894] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| AKR1C3 in Human [GtoPdb: 1382] [UniProtKB: P42330] | ||||||||
| GtoPdb | Determined in a competitive ABPP assay | - | 7.46 | pIC50 | 35 | nM | IC50 | J Med Chem (2025) 68: 9465-9478 [PMID:40277220] |
| GtoPdb | Determined in HEK293T cells overexpressing AKR1C1 | - | 7.89 | pIC50 | 13 | nM | IC50 | J Med Chem (2025) 68: 9465-9478 [PMID:40277220] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
