eneboparatide [Ligand Id: 13815] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| PTH1 receptor in Human [GtoPdb: 331] [UniProtKB: Q03431] | ||||||||
| GtoPdb | Measuring radioligand displacement at the R0 (G protein-uncoupled) conformation of hPTH1R using the radioligand 125I-PTH(1–34) in the presence of GTPγS to block receptor-G protein coupling | - | 8.82 | pIC50 | 1.5 | nM | IC50 | J Bone Miner Res (2016) 31: 1405-12 [PMID:26865415] |
| GtoPdb | Measuring radioligand displacement at the RG (G protein-coupled) conformation of hPTH1R using the radioligand 125I-M-PTH(1–15) | - | 10 | pIC50 | 0.1 | nM | IC50 | J Bone Miner Res (2016) 31: 1405-12 [PMID:26865415] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
