BI-43 [Ligand Id: 13398] activity data from GtoPdb

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  • glutaminyl-peptide cyclotransferase in Human [GtoPdb: 2411] [UniProtKB: Q16769]
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  • glutaminyl-peptide cyclotransferase like in Human [GtoPdb: 3289] [UniProtKB: Q9NXS2]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
glutaminyl-peptide cyclotransferase in Human [GtoPdb: 2411] [UniProtKB: Q16769]
GtoPdb - - 7.92 pIC50 12 nM IC50 J Med Chem (2024) 67: 8730-8756 [PMID:38817193]
glutaminyl-peptide cyclotransferase like in Human [GtoPdb: 3289] [UniProtKB: Q9NXS2]
GtoPdb - - 7.4 pIC50 40 nM IC50 J Med Chem (2024) 67: 8730-8756 [PMID:38817193]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.