iCARM1 [Ligand Id: 13358] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| coactivator associated arginine methyltransferase 1 in Human [GtoPdb: 1255] [UniProtKB: Q86X55] | ||||||||
| GtoPdb | Binding affinity determiend by SPR assay. | - | 6.17 | pKi | 678.5 | nM | Ki | J Med Chem (2024) 67: 7921-7934 [PMID:38713486] |
| GtoPdb | Inhibition of CARM1-mediated substrate peptide methylation in vitro. | - | 4.91 | pIC50 | 12300 | nM | IC50 | J Med Chem (2024) 67: 7921-7934 [PMID:38713486] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
