maridebart cafraglutide [Ligand Id: 13316] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GIP receptor in Monkey [GtoPdb: 248] | ||||||||
| GtoPdb | In vitro potency in GIPR recombinant cells | - | 7.58 | pIC50 | 26.5 | nM | IC50 | Nat Metab (2024) 6: 290-303 [PMID:38316982] |
| GIP receptor in Human [GtoPdb: 248] [UniProtKB: P48546] | ||||||||
| GtoPdb | In vitro potency in GIPR recombinant cells | - | 7.37 | pIC50 | 42.4 | nM | IC50 | Nat Metab (2024) 6: 290-303 [PMID:38316982] |
| GIP receptor in Rat [GtoPdb: 248] [UniProtKB: P43219] | ||||||||
| GtoPdb | In vitro potency in GIPR recombinant cells | - | 6.08 | pIC50 | 822.3 | nM | IC50 | Nat Metab (2024) 6: 290-303 [PMID:38316982] |
| GLP-1 receptor in Monkey [GtoPdb: 249] | ||||||||
| GtoPdb | In vitro potency in GLP-1R recombinant cells | - | 8.24 | pEC50 | 5.7 | nM | EC50 | Nat Metab (2024) 6: 290-303 [PMID:38316982] |
| GLP-1 receptor in Human [GtoPdb: 249] [UniProtKB: P43220] | ||||||||
| GtoPdb | In vitro potency in GLP-1R recombinant cells | - | 7.61 | pEC50 | 24.4 | nM | EC50 | Nat Metab (2024) 6: 290-303 [PMID:38316982] |
| GLP-1 receptor in Rat [GtoPdb: 249] [UniProtKB: P32301] | ||||||||
| GtoPdb | In vitro potency in GLP-1R recombinant cells | - | 8.62 | pEC50 | 2.4 | nM | EC50 | Nat Metab (2024) 6: 290-303 [PMID:38316982] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
