HS024 [Ligand Id: 1328] activity data from GtoPdb

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  • MC1 receptor in Human [GtoPdb: 282] [UniProtKB: Q01726]
Created with Highcharts 10.3.3ValuesChart context menuMC1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • MC3 receptor in Human [GtoPdb: 284] [UniProtKB: P41968]
Created with Highcharts 10.3.3ValuesChart context menuMC3 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • MC4 receptor in Human [GtoPdb: 285] [UniProtKB: P32245]
Created with Highcharts 10.3.3ValuesChart context menuMC4 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • MC5 receptor in Human [GtoPdb: 286] [UniProtKB: P33032]
Created with Highcharts 10.3.3ValuesChart context menuMC5 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
MC1 receptor in Human [GtoPdb: 282] [UniProtKB: Q01726]
GtoPdb - - 7.7 pKd - - - Endocrinology (1998) 139: 5006-14 [PMID:9832440]
MC3 receptor in Human [GtoPdb: 284] [UniProtKB: P41968]
GtoPdb - - 8.3 pKd - - - Endocrinology (1998) 139: 5006-14 [PMID:9832440]
MC4 receptor in Human [GtoPdb: 285] [UniProtKB: P32245]
GtoPdb - - 9.5 pKd - - - Endocrinology (1998) 139: 5006-14 [PMID:9832440]
MC5 receptor in Human [GtoPdb: 286] [UniProtKB: P33032]
GtoPdb - - 8.5 pKd - - - Endocrinology (1998) 139: 5006-14 [PMID:9832440]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.