CDN1163 [Ligand Id: 12968] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1474314
  • SERCA1 in Rabbit [GtoPdb: 840]
Created with Highcharts 10.3.3ValuesChart context menuSERCA1pKd RabbitpKi RabbitpIC50 RabbitpEC50 Rabbit0123456Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
SERCA1 in Rabbit [GtoPdb: 840]
GtoPdb Measuring enhanced Ca2+ ion translocation by SERCA ATP-ase in rabbit skeletal muscle SR vesicles that contain a high level of SERCA1a isoform - 5.22 pEC50 6000 nM EC50 ChemMedChem (2021) 16: 3293-3299 [PMID:34297466]

ChEMBL data shown on this page come from version 35:

Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]