I-287 [Ligand Id: 12491] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| PAR2 in Human [GtoPdb: 348] [UniProtKB: P55085] | ||||||||
| GtoPdb | Inhibition of Gα13 activation in hPAR2-HEK293 cells | - | 6.41 | pIC50 | 389 | nM | IC50 | Commun Biol (2020) 3: 719 [PMID:33247181] |
| GtoPdb | Inhibition of Gαq activation in hPAR2-HEK293 cells | - | 7.14 | pIC50 | 72.4 | nM | IC50 | Commun Biol (2020) 3: 719 [PMID:33247181] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
