compound 29 [PMID: 36356320] [Ligand Id: 12313] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362] | ||||||||
| GtoPdb | - | - | 7.68 | pIC50 | 21 | nM | IC50 | J Med Chem (2022) 65: 15433-15442 [PMID:36356320] |
| fibroblast growth factor receptor 2 in Human [GtoPdb: 1809] [UniProtKB: P21802] | ||||||||
| GtoPdb | - | - | 9 | pIC50 | 1 | nM | IC50 | J Med Chem (2022) 65: 15433-15442 [PMID:36356320] |
| fibroblast growth factor receptor 3 in Human [GtoPdb: 1810] [UniProtKB: P22607] | ||||||||
| GtoPdb | Inhibition of FGFR3V555L in vitro. | - | 8.57 | pIC50 | 2.7 | nM | IC50 | J Med Chem (2022) 65: 15433-15442 [PMID:36356320] |
| GtoPdb | Inhibition of WT FGFR3 in vitro. | - | 9.3 | pIC50 | 0.5 | nM | IC50 | J Med Chem (2022) 65: 15433-15442 [PMID:36356320] |
| fibroblast growth factor receptor 4 in Human [GtoPdb: 1811] [UniProtKB: P22455] | ||||||||
| GtoPdb | - | - | 6.84 | pIC50 | 145 | nM | IC50 | J Med Chem (2022) 65: 15433-15442 [PMID:36356320] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
