burimamide [Ligand Id: 1229] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| H2 receptor in Human [GtoPdb: 263] [UniProtKB: P25021] | ||||||||
| GtoPdb | - | - | 5.7 | pEC50 | - | - | - | J Neurochem (1998) 71: 799-807 [PMID:9681472] |
| H2 receptor in Rat [GtoPdb: 263] [UniProtKB: P25102] | ||||||||
| GtoPdb | - | - | 5.5 | pKi | - | - | - | Proc Natl Acad Sci USA (1996) 93: 6802-7 [PMID:8692899] |
| H3 receptor in Human [GtoPdb: 264] [UniProtKB: Q9Y5N1] | ||||||||
| GtoPdb | - | - | 7.1 | pKi | - | - | - |
J Pharmacol Exp Ther (2001) 299: 908-14 [PMID:11714875]; Mol Pharmacol (2001) 59: 420-6 [PMID:11179434] |
| H3 receptor in Rat [GtoPdb: 264] [UniProtKB: Q9QYN8] | ||||||||
| GtoPdb | - | - | 7.3 | pKi | - | - | - | J Pharmacol Exp Ther (2001) 299: 908-14 [PMID:11714875] |
| H4 receptor in Human [GtoPdb: 265] [UniProtKB: Q9H3N8] | ||||||||
| GtoPdb | - | - | 7.4 | pKi | - | - | - |
Mol Pharmacol (2001) 59: 420-6 [PMID:11179434]; J Pharmacol Exp Ther (2001) 299: 121-30 [PMID:11561071]; J Pharmacol Exp Ther (2001) 296: 1058-66 [PMID:11181941]; Mol Pharmacol (2001) 59: 434-41 [PMID:11179436]; J Pharmacol Exp Ther (2005) 314: 1310-21 [PMID:15947036] |
| H4 receptor in Mouse [GtoPdb: 265] [UniProtKB: Q91ZY2] | ||||||||
| GtoPdb | - | - | 6.1 | pKi | - | - | - | J Pharmacol Exp Ther (2001) 299: 121-30 [PMID:11561071] |
| H4 receptor in Rat [GtoPdb: 265] [UniProtKB: Q91ZY1] | ||||||||
| GtoPdb | - | - | 6 | pKi | - | - | - | J Pharmacol Exp Ther (2001) 299: 121-30 [PMID:11561071] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
