upacicalcet [Ligand Id: 12235] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| CaS receptor in Human [GtoPdb: 54] [UniProtKB: P41180] | ||||||||
| GtoPdb | Competition binding assay, dispalcement of [3H]-upacicalcet from hCaSR by unlabelled upacicalcet | - | 8.09 | pIC50 | 8.2 | nM | IC50 | Mol Pharmacol (2022) 102: 183-195 [PMID:36122913] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
