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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference | 
|---|---|---|---|---|---|---|---|---|
| protein kinase, membrane associated tyrosine/threonine 1 in Human [GtoPdb: 2167] [UniProtKB: Q99640] | ||||||||
| GtoPdb | Determined in a NanoBRET target engagement assay | - | 8.7 | pIC50 | 2 | nM | IC50 | J Med Chem (2022) 65: 10251-10284 [PMID:35880755] | 
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.