JX35 [Ligand Id: 11945] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Plasmodium falciparum histone deacetylase 1 in Plasmodium falciparum NF54 [GtoPdb: 3072] | ||||||||
| GtoPdb | Parasite early stage (II) gametocyte assay | - | 7.8 | pIC50 | 15.83 | nM | IC50 | J Med Chem (2022) 65: 4156-4181 [PMID:35175762] |
| GtoPdb | Parasite late stage (V) gametocyte assay | - | 7.91 | pIC50 | 12.42 | nM | IC50 | J Med Chem (2022) 65: 4156-4181 [PMID:35175762] |
| Plasmodium falciparum histone deacetylase 1 in Plasmodium falciparum 3D7 [GtoPdb: 3072] [UniProtKB: Q7K6A1] | ||||||||
| GtoPdb | Parasite growth inhibition assay | - | 8.9 | pIC50 | 1.26 | nM | IC50 | J Med Chem (2022) 65: 4156-4181 [PMID:35175762] |
| Plasmodium falciparum histone deacetylase 1 in Plasmodium falciparum Dd2 [GtoPdb: 3072] | ||||||||
| GtoPdb | Parasite growth inhibition assay | - | 8.79 | pIC50 | 1.61 | nM | IC50 | J Med Chem (2022) 65: 4156-4181 [PMID:35175762] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
