compound 17b [PMID: 35286086] [Ligand Id: 11941] activity data from GtoPdb

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  • Estrogen receptor-α in Human [GtoPdb: 620] [UniProtKB: P03372]
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  • epidermal growth factor receptor in Human [GtoPdb: 1797] [UniProtKB: P00533]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Estrogen receptor-α in Human [GtoPdb: 620] [UniProtKB: P03372]
GtoPdb - - 8.34 pIC50 4.6 nM IC50 J Med Chem (2022) 65: 4616-4632 [PMID:35286086]
epidermal growth factor receptor in Human [GtoPdb: 1797] [UniProtKB: P00533]
GtoPdb - - 8.6 pIC50 2.5 nM IC50 J Med Chem (2022) 65: 4616-4632 [PMID:35286086]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.