compound 13 [PMID: 34333981] [Ligand Id: 11895] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • AP2 associated kinase 1 in Human [GtoPdb: 1921] [UniProtKB: Q2M2I8]
There should be some charts here, you may need to enable JavaScript!
  • BMP2 inducible kinase in Human [GtoPdb: 1941] [UniProtKB: Q9NSY1]
There should be some charts here, you may need to enable JavaScript!
  • serine/threonine kinase 16 in Human [GtoPdb: 2213] [UniProtKB: O75716]
There should be some charts here, you may need to enable JavaScript!
  • tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
AP2 associated kinase 1 in Human [GtoPdb: 1921] [UniProtKB: Q2M2I8]
GtoPdb - - 7.13 pIC50 74 nM IC50 J Med Chem (2022) 65: 1313-1328 [PMID:34333981]
BMP2 inducible kinase in Human [GtoPdb: 1941] [UniProtKB: Q9NSY1]
GtoPdb - - 7.4 pIC50 40 nM IC50 J Med Chem (2022) 65: 1313-1328 [PMID:34333981]
serine/threonine kinase 16 in Human [GtoPdb: 2213] [UniProtKB: O75716]
GtoPdb - - 7.09 pIC50 82 nM IC50 J Med Chem (2022) 65: 1313-1328 [PMID:34333981]
tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597]
GtoPdb - - 7.32 pIC50 48 nM IC50 J Med Chem (2022) 65: 1313-1328 [PMID:34333981]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.