bezuclastinib [Ligand Id: 11868] activity data from GtoPdb

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  • KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721]
GtoPdb Inhibition of KITV560G/D816V - 7.55 pIC50 28 nM IC50 Clin Exp Med (2019) 19: 201-210 [PMID:30523507]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.