IMP-1002 [Ligand Id: 11850] activity data from GtoPdb

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  • Plasmodium falciparum N-myristoyltransferase in Plasmodium falciparum 3D7 [GtoPdb: 2955] [UniProtKB: Q8ILW6]
  • Plasmodium falciparum N-myristoyltransferase in Plasmodium falciparum Dd2 [GtoPdb: 2955]
Created with Highcharts 10.3.3ValuesChart context menuPlasmodium falciparum N-myristoyltransferasepKd Plasmodiumfalciparum 3D7pKi Plasmodiumfalciparum 3D7pIC50 Plasmodiumfalciparum 3D7pEC50 Plasmodiumfalciparum 3D7pKd Plasmodiumfalciparum Dd2pKi Plasmodiumfalciparum Dd2pIC50 Plasmodiumfalciparum Dd2pEC50 Plasmodiumfalciparum Dd20246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Plasmodium falciparum N-myristoyltransferase in Plasmodium falciparum 3D7 [GtoPdb: 2955] [UniProtKB: Q8ILW6]
GtoPdb Parasite growth inhibition assay - 7.47 pEC50 34 nM EC50 Cell Chem Biol (2019) 26: 991-1000.e7 [PMID:31080074]
Plasmodium falciparum N-myristoyltransferase in Plasmodium falciparum Dd2 [GtoPdb: 2955]
GtoPdb Parasite growth inhibition assay - 7.69 pEC50 20.4 nM EC50 Cell Chem Biol (2019) 26: 991-1000.e7 [PMID:31080074]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.