BPR1R024 [Ligand Id: 11747] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| platelet derived growth factor receptor alpha in Human [GtoPdb: 1803] [UniProtKB: P16234] | ||||||||
| GtoPdb | - | - | 7.28 | pIC50 | 52.7 | nM | IC50 | J Med Chem (2021) 64: 14477-14497 [PMID:34606263] |
| platelet derived growth factor receptor beta in Human [GtoPdb: 1804] [UniProtKB: P09619] | ||||||||
| GtoPdb | - | - | 7.5 | pIC50 | 31.5 | nM | IC50 | J Med Chem (2021) 64: 14477-14497 [PMID:34606263] |
| KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721] | ||||||||
| GtoPdb | - | - | 8.96 | pIC50 | 1.1 | nM | IC50 | J Med Chem (2021) 64: 14477-14497 [PMID:34606263] |
| colony stimulating factor 1 receptor in Human [GtoPdb: 1806] [UniProtKB: P07333] | ||||||||
| GtoPdb | - | - | 9.28 | pIC50 | 0.53 | nM | IC50 | J Med Chem (2021) 64: 14477-14497 [PMID:34606263] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
