vepafestinib [Ligand Id: 11678] activity data from GtoPdb

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  • ret proto-oncogene in Human [GtoPdb: 2185] [UniProtKB: P07949]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
ret proto-oncogene in Human [GtoPdb: 2185] [UniProtKB: P07949]
GtoPdb Inhibition of peptide substrate phosphorylation by recombinant human RET in the presence of test compound - 9.7 pIC50 0.2 nM IC50 US20180009818A1. Novel fused pyrimidine compound or salt thereof (2018)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.