SD-91 [Ligand Id: 11599] activity data from GtoPdb

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  • signal transducer and activator of transcription 3 in Human [GtoPdb: 2994] [UniProtKB: P40763]
Created with Highcharts 10.3.3ValuesChart context menusignal transducer and activator of transcription 3pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
signal transducer and activator of transcription 3 in Human [GtoPdb: 2994] [UniProtKB: P40763]
GtoPdb Determined in a biolayer interferometry (BLI) assay - 7.55 pKd 28 nM Kd ACS Med Chem Lett (2021) 12: 996-1004 [PMID:34141084]
GtoPdb Determined in a competitive fluorescence-polarization assay - 8.26 pKi 5.5 nM Ki ACS Med Chem Lett (2021) 12: 996-1004 [PMID:34141084]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.