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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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peptidylprolyl cis/trans isomerase, NIMA-interacting 1 in Human [GtoPdb: 3171] [UniProtKB: Q13526] | ||||||||
GtoPdb | Inhibition of Pin1 catalytic activity determined in a chymotrypsin-coupled peptidyl-prolyl isomerization assay (PPIase) assay | - | 6.68 | pKi | 211 | nM | Ki | Nat Chem Biol (2021) 17: 954-963 [PMID:33972797] |
GtoPdb | Binding to Pin1 in a fluorescence polarization (FP) assay that measured competitive displacement of an N-terminal fluorescein-labeled peptide substrate (Bth-D-pThr-Pip-Nal) | - | 7.77 | pKi | 17 | nM | Ki | Nat Chem Biol (2021) 17: 954-963 [PMID:33972797] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.