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ChEMBL ligand: CHEMBL1088750 (ARRY-371797, Arry-797, ARRY-797) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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mitogen-activated protein kinase 14/MAP kinase p38 alpha in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL260] [GtoPdb: 1499] [UniProtKB: Q16539] | ||||||||
ChEMBL | Inhibition of human recombinant p38alpha by liquid scintillation counting | B | 8.35 | pIC50 | 4.5 | nM | IC50 | J. Med. Chem. (2010) 53: 2345-2353 [PMID:19950901] |
GtoPdb | In vitro enzyme inhibition assay. | - | 8.35 | pIC50 | 4.5 | nM | IC50 | J Med Chem (2010) 53: 2345-53 [PMID:19950901] |
ChEMBL data shown on this page come from version 31:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]