compound 15 [PMID: 32045236] [Ligand Id: 10706] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Ecto-5'-Nucleotidase in Human [GtoPdb: 1232] [UniProtKB: P21589] | ||||||||
| GtoPdb | Ki vs. soluble human CD73 in vitro. | - | 8.44 | pKi | 3.59 | nM | Ki | J Med Chem (2020) 63: 2941-2957 [PMID:32045236] |
| GtoPdb | Inhibition of CD73 in human MDA-MB-231 cancer cells. | - | 8.48 | pKi | 3.33 | nM | Ki | J Med Chem (2020) 63: 2941-2957 [PMID:32045236] |
| Ecto-5'-Nucleotidase in Rat [GtoPdb: 1232] [UniProtKB: P21588] | ||||||||
| GtoPdb | Ki vs. soluble rat CD73 in vitro. | - | 7.82 | pKi | 15.1 | nM | Ki | J Med Chem (2020) 63: 2941-2957 [PMID:32045236] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
