compound 5 [Tomassi et al., 2020] [Ligand Id: 10672] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| poly(ADP-ribose) polymerase 1 in Human [GtoPdb: 2771] [UniProtKB: P09874] | ||||||||
| GtoPdb | - | - | 7.05 | pIC50 | 89.6 | nM | IC50 | ACS Med Chem Lett (2020) : |
| poly(ADP-ribose) polymerase 2 in Human [GtoPdb: 2772] [UniProtKB: Q9UGN5] | ||||||||
| GtoPdb | - | - | 7.42 | pIC50 | 37.8 | nM | IC50 | ACS Med Chem Lett (2020) : |
| tankyrase in Human [GtoPdb: 3108] [UniProtKB: O95271] | ||||||||
| GtoPdb | - | - | 8.21 | pIC50 | 6.1 | nM | IC50 | ACS Med Chem Lett (2020) : |
| tankyrase 2 in Human [GtoPdb: 3109] [UniProtKB: Q9H2K2] | ||||||||
| GtoPdb | - | - | 9.52 | pIC50 | 0.3 | nM | IC50 | ACS Med Chem Lett (2020) : |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
