UCSF7447 [Ligand Id: 10666] activity data from GtoPdb

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  • MT1 receptor in Human [GtoPdb: 287] [UniProtKB: P48039]
Created with Highcharts 10.3.3ValuesChart context menuMT1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • MT2 receptor in Human [GtoPdb: 288] [UniProtKB: P49286]
Created with Highcharts 10.3.3ValuesChart context menuMT2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human01234567Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
MT1 receptor in Human [GtoPdb: 287] [UniProtKB: P48039]
GtoPdb - - 7.32 pEC50 47.86 nM EC50 Nature (2020) 579: 609-614 [PMID:32040955]
MT2 receptor in Human [GtoPdb: 288] [UniProtKB: P49286]
GtoPdb - - 5.99 pEC50 1023.9 nM EC50 Nature (2020) 579: 609-614 [PMID:32040955]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.