compound 25 [Zhang et al., 2020] [Ligand Id: 10643] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| RAR-related orphan receptor-γ in Human [GtoPdb: 600] [UniProtKB: P51449] | ||||||||
| GtoPdb | Inhibition of cofactor (LXXLL-motif containing steroid receptor coactivator SRC1 peptide) recruitment to RORγ ligand binding domain in a TR-FRET biochemical assay. | - | 9 | pIC50 | 1 | nM | IC50 | ACS Med Chem Lett (2020) 11: 114-119 [PMID:32071676] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
