itacnosertib [Ligand Id: 10632] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| activin A receptor type 1 in Human [GtoPdb: 1785] [UniProtKB: Q04771] | ||||||||
| GtoPdb | Inhibitory activity against human AKL2, determined using a LanthaScreen® binding assay. | - | 8 | pIC50 | <10 | nM | IC50 | WO2014151871A9. Jak2 and alk2 inhibitors and methods for their use (2014) |
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | Inhibitory activity against human JAK2 kinase, determined using a Z'-Lyte® biochemical assay. | - | 6 | pIC50 | >1000 | nM | IC50 | WO2014151871A9. Jak2 and alk2 inhibitors and methods for their use (2014) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
