uzansertib [Ligand Id: 10626] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Pim-1 proto-oncogene, serine/threonine kinase in Human [GtoPdb: 2158] [UniProtKB: P11309] | ||||||||
| GtoPdb | Kinase inhibition in a biochemical enzyme activity assay. | - | 9.62 | pIC50 | 0.24 | nM | IC50 | PLoS ONE (2018) 13: e0199108 [PMID:29927999] |
| Pim-2 proto-oncogene, serine/threonine kinase in Human [GtoPdb: 2159] [UniProtKB: Q9P1W9] | ||||||||
| GtoPdb | Kinase inhibition in a biochemical enzyme activity assay. | - | 7.52 | pIC50 | 30 | nM | IC50 | PLoS ONE (2018) 13: e0199108 [PMID:29927999] |
| Pim-3 proto-oncogene, serine/threonine kinase in Human [GtoPdb: 2160] [UniProtKB: Q86V86] | ||||||||
| GtoPdb | Kinase inhibition in a biochemical enzyme activity assay. | - | 9.92 | pIC50 | 0.12 | nM | IC50 | PLoS ONE (2018) 13: e0199108 [PMID:29927999] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
