balovaptan [Ligand Id: 10615] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| 5-HT2B receptor in Human [GtoPdb: 7] [UniProtKB: P41595] | ||||||||
| GtoPdb | - | - | 11.57 | pKd | 0 | nM | Kd | J Med Chem (2020) 63: 1511-1525 [PMID:31951127] |
| V1A receptor in Human [GtoPdb: 366] [UniProtKB: P37288] | ||||||||
| GtoPdb | - | - | 8.59 | pKd | 2.56 | nM | Kd | J Med Chem (2020) 63: 1511-1525 [PMID:31951127] |
| V2 receptor in Human [GtoPdb: 368] [UniProtKB: P30518] | ||||||||
| GtoPdb | - | - | 5 | pKd | 9953 | nM | Kd | J Med Chem (2020) 63: 1511-1525 [PMID:31951127] |
| OT receptor in Human [GtoPdb: 369] [UniProtKB: P30559] | ||||||||
| GtoPdb | - | - | 5.15 | pKi | 7002 | nM | Ki | J Med Chem (2020) 63: 1511-1525 [PMID:31951127] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
