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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GPR15 in Human [GtoPdb: 87] [UniProtKB: P49685] | ||||||||
| GtoPdb | Agonist activity determined in vitro, measuring calcium response in CHO-K1 cells expressing hGPR15 and Aequorin. | - | 5.85 | pEC50 | 1400 | nM | EC50 | Sci Signal (2017) 10: [PMID:28900043] |
| MRGPRX1 in Human [GtoPdb: 156] [UniProtKB: Q96LB2] | ||||||||
| GtoPdb | Determined in a FLIPR calcium imaging assay using HEK cells heterologously expressing hMRGPRX1 | - | 4.74 | pEC50 | 18100 | nM | EC50 | Sci Adv (2022) 8: eabm7342 [PMID:35704588] |
| MRGPRX2 in Human [GtoPdb: 157] [UniProtKB: Q96LB1] | ||||||||
| GtoPdb | Determined in a FLIPR calcium imaging assay using HEK cells heterologously expressing hMRGPRX2 | - | 5.72 | pEC50 | 1900 | nM | EC50 | Sci Adv (2022) 8: eabm7342 [PMID:35704588] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.