ARV-771 [Ligand Id: 10564] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| bromodomain containing 2 in Human [GtoPdb: 1944] [UniProtKB: P25440] | ||||||||
| GtoPdb | Binding affinity for bromodomain 2 of hBRD2. | - | 8.33 | pKd | 4.7 | nM | Kd | Proc Natl Acad Sci USA (2016) 113: 7124-9 [PMID:27274052] |
| bromodomain containing 4 in Human [GtoPdb: 1945] [UniProtKB: O60885] | ||||||||
| GtoPdb | Binding affinity for bromodomain 2 of hBRD4. | - | 8.12 | pKd | 7.6 | nM | Kd | Proc Natl Acad Sci USA (2016) 113: 7124-9 [PMID:27274052] |
| bromodomain containing 3 in Human [GtoPdb: 2725] [UniProtKB: Q15059] | ||||||||
| GtoPdb | Binding affinity for bromodomain 2 of hBRD3. | - | 8.12 | pKd | 7.6 | nM | Kd | Proc Natl Acad Sci USA (2016) 113: 7124-9 [PMID:27274052] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
