dBRD9 [Ligand Id: 10545] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| bromodomain containing 9 in Human [GtoPdb: 2728] [UniProtKB: Q9H8M2] | ||||||||
| GtoPdb | AlphaScreen competitive ligand binding assay using recombinant BRD9. | - | 6.98 | pIC50 | 104 | nM | IC50 | Angew Chem Int Ed Engl (2017) 56: 5738-5743 [PMID:28418626] |
| cereblon in Human [GtoPdb: 3086] [UniProtKB: Q96SW2] | ||||||||
| GtoPdb | AlphaScreen competitive ligand binding assay using the CRBN-DDB1 complex. | - | 7.5 | pIC50 | 31.3 | nM | IC50 | Angew Chem Int Ed Engl (2017) 56: 5738-5743 [PMID:28418626] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
