compound 1 [PMID: 31465224] [Ligand Id: 10493] activity data from GtoPdb

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  • pyruvate kinase M1/2 in Human [GtoPdb: 3006] [UniProtKB: P14618]
Created with Highcharts 10.3.3ValuesChart context menupyruvate kinase M1/2pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
pyruvate kinase M1/2 in Human [GtoPdb: 3006] [UniProtKB: P14618]
GtoPdb Measuring inhibition of pyruvate kinase activity in PC-9 cells treated with compound 1. - 6.6 pIC50 250 nM IC50 J Med Chem (2019) 62: 8497-8510 [PMID:31465224]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.