compound 5a [PMID: 31287314] [Ligand Id: 10433] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| carbonic anhydrase 1 in Human [GtoPdb: 2597] [UniProtKB: P00915] | ||||||||
| GtoPdb | - | - | 6.07 | pKi | 851.7 | nM | Ki | J Med Chem (2019) 62: 7233-7249 [PMID:31287314] |
| carbonic anhydrase 4 in Human [GtoPdb: 2599] [UniProtKB: P22748] | ||||||||
| GtoPdb | - | - | 5 | pKi | >10000 | nM | Ki | J Med Chem (2019) 62: 7233-7249 [PMID:31287314] |
| carbonic anhydrase 12 in Human [GtoPdb: 2747] [UniProtKB: O43570] | ||||||||
| GtoPdb | - | - | 6.11 | pKi | 783.8 | nM | Ki | J Med Chem (2019) 62: 7233-7249 [PMID:31287314] |
| carbonic anhydrase 9 in Human [GtoPdb: 3055] [UniProtKB: Q16790] | ||||||||
| GtoPdb | - | - | 6.38 | pKi | 415.9 | nM | Ki | J Med Chem (2019) 62: 7233-7249 [PMID:31287314] |
| carbonic anhydrase 2 in Human [GtoPdb: 3092] [UniProtKB: P00918] | ||||||||
| GtoPdb | - | - | 7.02 | pKi | 96.5 | nM | Ki | J Med Chem (2019) 62: 7233-7249 [PMID:31287314] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
