AM237 [Ligand Id: 10421] activity data from GtoPdb

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  • TRPC5 in Human [GtoPdb: 490] [UniProtKB: Q9UL62]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TRPC5 in Human [GtoPdb: 490] [UniProtKB: Q9UL62]
GtoPdb EC50 determined in HEK T-REx cells over-expressing homomeric TRPC5 channels, by measuring ligand-induced modulation of intracellular Ca2+. - 7.7 pEC50 20 nM EC50 Br J Pharmacol (2019) 176: 3924-3938 [PMID:31277085]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.