GI‐530159 [Ligand Id: 10337] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| K2P2.1 in Human [GtoPdb: 514] [UniProtKB: O95069] | ||||||||
| GtoPdb | Measuring GI‐530139-induced enhanced current via single hTREK1 channels measured at +60 mV in the inside‐out manual patch configuration, in a concentration–response experiment. | - | 6.05 | pEC50 | 890 | nM | EC50 | Br J Pharmacol (2018) 175: 2272-2283 [PMID:29150838] |
| GtoPdb | Measuring 86Rb efflux by TREK1 induced by GI‐530159 at 70 mM potassium. | - | 6.12 | pEC50 | 760 | nM | EC50 | Br J Pharmacol (2018) 175: 2272-2283 [PMID:29150838] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
