compound 3f [Festa et al., 2019] [Ligand Id: 10187] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Farnesoid X receptor in Human [GtoPdb: 603] [UniProtKB: Q96RI1] | ||||||||
| GtoPdb | Cellular potency (HepG2 cells) measured as antagonism of CDCA-induced FXR activation in a transactivation reporter assay. | - | 6.24 | pIC50 | 580 | nM | IC50 | ACS Med Chem Lett (2019) 10: 504-510 [PMID:30996787] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
