compound 28 [Heitel et al., 2019] [Ligand Id: 10186] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Retinoid X receptor-α in Human [GtoPdb: 610] [UniProtKB: P19793] | ||||||||
| GtoPdb | In a cell-free isothermal titration calorimetry (ITC) assay. | - | 7.02 | pKd | 95 | nM | Kd | ACS Med Chem Lett (2019) 10: 203-208 [PMID:30783504] |
| GtoPdb | In a whole cell reporter gene assay. | - | 6.55 | pEC50 | 280 | nM | EC50 | ACS Med Chem Lett (2019) 10: 203-208 [PMID:30783504] |
| Retinoid X receptor-β in Human [GtoPdb: 611] [UniProtKB: P28702] | ||||||||
| GtoPdb | - | - | 6.51 | pEC50 | 310 | nM | EC50 | ACS Med Chem Lett (2019) 10: 203-208 [PMID:30783504] |
| Retinoid X receptor-γ in Human [GtoPdb: 612] [UniProtKB: P48443] | ||||||||
| GtoPdb | - | - | 5.8 | pEC50 | 1600 | nM | EC50 | ACS Med Chem Lett (2019) 10: 203-208 [PMID:30783504] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
