7-BIA [Ligand Id: 10109] activity data from GtoPdb

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  • RTP Type D in Human [GtoPdb: 1853] [UniProtKB: P23468]
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  • RTP Type S in Human [GtoPdb: 1866] [UniProtKB: Q13332]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
RTP Type D in Human [GtoPdb: 1853] [UniProtKB: P23468]
GtoPdb Inhibition of p-nitrophenyl phosphate dephosphorylation by recombinant PTPRD phosphatase domain fusion protein following 16-18 minute preincubation. - 6 pIC50 1000 nM IC50 Proc Natl Acad Sci USA (2018) 115: 11597-11602 [PMID:30348770]
RTP Type S in Human [GtoPdb: 1866] [UniProtKB: Q13332]
GtoPdb Inhibition of p-nitrophenyl phosphate dephosphorylation by recombinant PTPRS phosphatase domain fusion protein following 16-18 minute preincubation. - 4.4 pIC50 40000 nM IC50 J Clin Invest (1997) 100: 1137-43 [PMID:9276730]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.