setogepram [Ligand Id: 10043] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GPR84 in Human [GtoPdb: 120] [UniProtKB: Q9NQS5] | ||||||||
| GtoPdb | Measuring antagonist-dependent inhibition of Gαiactivation by sodium decanoate (agonist) in receptor transfected HEK293 cells. | - | 3.4 | pIC50 | 398107 | nM | IC50 | Am J Pathol (2018) 188: 1132-1148 [PMID:29454750] |
| FFA1 receptor in Human [GtoPdb: 225] [UniProtKB: O14842] | ||||||||
| GtoPdb | In a β-arrestin 2 recruitment assay measured by BRET. | - | 2.98 | pEC50 | 1047129 | nM | EC50 | Am J Pathol (2018) 188: 1132-1148 [PMID:29454750] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
