VU0483605 [Ligand Id: 10009] activity data from GtoPdb

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  • mGlu1 receptor in Human [GtoPdb: 289] [UniProtKB: Q13255]
Created with Highcharts 10.3.3ValuesChart context menumGlu1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • mGlu5 receptor in Rat [GtoPdb: 293] [UniProtKB: P31424]
Created with Highcharts 10.3.3ValuesChart context menumGlu5 receptorpKd RatpKi RatpIC50 RatpEC50 Rat0Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
mGlu1 receptor in Human [GtoPdb: 289] [UniProtKB: Q13255]
GtoPdb - - 6.41 pEC50 390 nM EC50 ACS Chem Biol (2014) 9: 2334-46 [PMID:25137254]
mGlu5 receptor in Rat [GtoPdb: 293] [UniProtKB: P31424]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.