Organic cation transporters (OCT) are electrogenic, Na⁺-independent and reversible.

Corticosterone and quinine are able to inhibit all three organic cation transporters.

* Key recommended reading is highlighted with an asterisk

* A-González N, Castrillo A. (2011) Liver X receptors as regulators of macrophage inflammatory and metabolic pathways. Biochim. Biophys. Acta, 1812 (8): 982-94. [PMID:21193033]

* Koepsell H. (2013) The SLC22 family with transporters of organic cations, anions and zwitterions. Mol. Aspects Med., 34 (2-3): 413-35. [PMID:23506881]

* Lozano E, Herraez E, Briz O, Robledo VS, Hernandez-Iglesias J, Gonzalez-Hernandez A, Marin JJ. (2013) Role of the plasma membrane transporter of organic cations OCT1 and its genetic variants in modern liver pharmacology. Biomed Res Int, 2013: 692071. [PMID:23984399]

* Pelis RM, Wright SH. (2014) SLC22, SLC44, and SLC47 transporters--organic anion and cation transporters: molecular and cellular properties. Curr Top Membr, 73: 233-61. [PMID:24745985]

* Yin J, Wang J. (2016) Renal drug transporters and their significance in drug-drug interactions. Acta Pharm Sin B, 6 (5): 363-373. [PMID:27709005]

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