GtoPdb is requesting financial support from commercial users. Please see our sustainability page for more information.

R-486   Click here for help

GtoPdb Ligand ID: 2105

Synonyms: [Trp7,β-Ala8]neurokinin A(4-10) | MEN 10295 | R 486 | R486
Compound class: Peptide
Click here for help
Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
NK1 receptor Hs Antagonist Antagonist 6.5 – 6.6 pKi - 1
pKi 6.5 – 6.6 [1]