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Unless otherwise stated all data on this page refer to the human proteins. Gene information is provided for human (Hs), mouse (Mm) and rat (Rn).
ASH1 like histone lysine methyltransferase Show summary »« Hide summary
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DOT1 like histone lysine methyltransferase Show summary »« Hide summary More detailed page
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euchromatic histone lysine methyltransferase 1 Show summary »« Hide summary
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euchromatic histone lysine methyltransferase 2 Show summary »« Hide summary
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EZH1 (enhancer of zeste 1 polycomb repressive complex 2 subunit) Show summary »« Hide summary More detailed page
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EZH2 (enhancer of zeste 2 polycomb repressive complex 2 subunit) Show summary »« Hide summary More detailed page
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lysine methyltransferase 2B Show summary »« Hide summary
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lysine methyltransferase 2A Show summary »« Hide summary
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lysine methyltransferase 2C Show summary »« Hide summary
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lysine methyltransferase 2D Show summary »« Hide summary
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lysine methyltransferase 2E (inactive) Show summary »« Hide summary
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lysine methyltransferase 5A Show summary »« Hide summary
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lysine methyltransferase 5B Show summary »« Hide summary
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lysine methyltransferase 5C Show summary »« Hide summary
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nuclear receptor binding SET domain protein 1 Show summary »« Hide summary
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nuclear receptor binding SET domain protein 2 Show summary »« Hide summary
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PR/SET domain 2 Show summary »« Hide summary
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SET domain containing 1A, histone lysine methyltransferase Show summary »« Hide summary
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SET domain containing 1B, histone lysine methyltransferase Show summary »« Hide summary
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SET domain containing 2, histone lysine methyltransferase Show summary »« Hide summary
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SET domain containing 7, histone lysine methyltransferase Show summary »« Hide summary More detailed page
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SET domain bifurcated histone lysine methyltransferase 1 Show summary »« Hide summary
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SET domain bifurcated histone lysine methyltransferase 2 Show summary »« Hide summary
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SET and MYND domain containing 2 Show summary »« Hide summary More detailed page
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SUV39H1 histone lysine methyltransferase Show summary »« Hide summary
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SUV39H2 histone lysine methyltransferase Show summary »« Hide summary
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32. SGC. A-366: a chemical Probe for G9a/GLP. Accessed on 03/03/2015. Modified on 04/08/2023. thesgc.org, https://www.thesgc.org/chemical-probes/A-366
33. SGC. LLY-507: A chemical probe for SMYD2 protein lysine methyltransferase. Accessed on 03/03/2015. Modified on 04/08/2023. thesgc.org, https://www.thesgc.org/chemical-probes/LLY-507
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Database page citation:
2.1.1.43 Histone methyltransferases (HMTs). Accessed on 04/11/2024. IUPHAR/BPS Guide to PHARMACOLOGY, http://www.guidetopharmacology.org/GRAC/FamilyDisplayForward?familyId=871.
Concise Guide to PHARMACOLOGY citation:
Alexander SPH, Fabbro D, Kelly E, Mathie AA, Peters JA, Veale EL, Armstrong JF, Faccenda E, Harding SD, Davies JA et al. (2023) The Concise Guide to PHARMACOLOGY 2023/24: Enzymes. Br J Pharmacol. 180 Suppl 2:S289-373.
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