CCT196969 [Ligand Id: 9815] activity data from GtoPdb

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  • B-Raf proto-oncogene, serine/threonine kinase in Human [GtoPdb: 1943] [UniProtKB: P15056]
  • This target only has 0 pki data point
  • 0
1 _lig_chart_1 B-Raf proto-oncogene, serine/threonine kinase Human
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  • LCK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2053] [UniProtKB: P06239]
  • This target only has 0 pki data point
  • 0
2 _lig_chart_2 LCK proto-oncogene, Src family tyrosine kinase Human
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  • Raf-1 proto-oncogene, serine/threonine kinase in Human [GtoPdb: 2184] [UniProtKB: P04049]
  • This target only has 0 pki data point
  • 0
3 _lig_chart_3 Raf-1 proto-oncogene, serine/threonine kinase Human
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  • SRC proto-oncogene, non-receptor tyrosine kinase in Human [GtoPdb: 2206] [UniProtKB: P12931]
  • This target only has 0 pki data point
  • 0
4 _lig_chart_4 SRC proto-oncogene, non-receptor tyrosine kinase Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
B-Raf proto-oncogene, serine/threonine kinase in Human [GtoPdb: 1943] [UniProtKB: P15056]
GtoPdb - - 7 pIC50 100 nM IC50 Cancer Cell (2015) 27: 85-96 [PMID:25500121]
LCK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2053] [UniProtKB: P06239]
GtoPdb - - 7.7 pIC50 20 nM IC50 Cancer Cell (2015) 27: 85-96 [PMID:25500121]
Raf-1 proto-oncogene, serine/threonine kinase in Human [GtoPdb: 2184] [UniProtKB: P04049]
GtoPdb - - 8 pIC50 10 nM IC50 Cancer Cell (2015) 27: 85-96 [PMID:25500121]
SRC proto-oncogene, non-receptor tyrosine kinase in Human [GtoPdb: 2206] [UniProtKB: P12931]
GtoPdb - - 7.52 pIC50 30 nM IC50 Cancer Cell (2015) 27: 85-96 [PMID:25500121]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.