GNE-3500 [Ligand Id: 9660] activity data from GtoPdb

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  • RAR-related orphan receptor-γ in Human [GtoPdb: 600] [UniProtKB: P51449]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
RAR-related orphan receptor-γ in Human [GtoPdb: 600] [UniProtKB: P51449]
GtoPdb Measuring inhibition of SRC1 coactivator peptide recruitment by the ligand binding domain of human RORγ. - 7.92 pEC50 12 nM EC50 J Med Chem (2015) 58: 5308-22 [PMID:26061388]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.