ritlecitinib [Ligand Id: 9559] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Janus kinase 1 in Human [GtoPdb: 2047] [UniProtKB: P23458] | ||||||||
| GtoPdb | At 1 mM ATP. | - | 5.79 | pIC50 | 1640 | nM | IC50 | J Med Chem (2017) 60: 1971-1993 [PMID:28139931] |
| Janus kinase 3 in Human [GtoPdb: 2049] [UniProtKB: P52333] | ||||||||
| GtoPdb | At 4 μM ATP (Km). | - | 9.52 | pIC50 | 0.3 | nM | IC50 | |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
