ChEMBL ligand: CHEMBL1215923 (Bimosiamose, TBC-1269)
selectin P (CD62)/P-selectin in Human [ChEMBL: CHEMBL5378] [GtoPdb: 3103] [UniProtKB: P16109] There should be some charts here, you may need to enable JavaScript!
P-selectin glycoprotein ligand 1 in Human [ChEMBL: CHEMBL4183] [UniProtKB: Q14242] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
selectin P (CD62)/P-selectin in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5378] [GtoPdb: 3103] [UniProtKB: P16109]
ChEMBL	Inhibition of human P-selectin after 2 hrs	B	4.02	pIC50	95000	nM	IC50	J Med Chem (2007) 50: 1101-1115 [PMID:17302397]
GtoPdb	Inhibition of P-selectin binding in an HL-60 cellular assay.	-	4.15	pIC50	70000	nM	IC50	J Med Chem (1998) 41: 1099-111 [PMID:9544210]
ChEMBL	Inhibition of P-selectin in human HL-60 cells	B	4.15	pIC50	70000	nM	IC50	J Med Chem (2010) 53: 6003-6017 [PMID:20718494]
P-selectin glycoprotein ligand 1 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4183] [UniProtKB: Q14242]
ChEMBL	Inhibition of P-selectin-mediated adhesion of HL60 cells	B	4.15	pIC50	70000	nM	IC50	J Med Chem (2007) 50: 21-39 [PMID:17201408]

ChEMBL data shown on this page come from version 32:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]