quinostatin [Ligand Id: 8978] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336] | ||||||||
| GtoPdb | In vitro binding affinity to recombinant complex of PI3K alpha regulatory and catalytic subunits. | - | 6.22 | pKd | 600 | nM | Kd | Chem Biol (2007) 14: 371-7 [PMID:17462572] |
| GtoPdb | Inhibition of lipid-kinase activity in vitro. | - | 4.82 | pIC50 | 15000 | nM | IC50 | Chem Biol (2007) 14: 371-7 [PMID:17462572] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736] | ||||||||
| GtoPdb | Inhibition of lipid-kinase activity in vitro. | - | 4.52 | pIC50 | 30000 | nM | IC50 | Chem Biol (2007) 14: 371-7 [PMID:17462572] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
